TITLE

Bioisosterism: A Useful Strategy for Molecular Modification and Drug Design

AUTHOR(S)
Lima, L�dia Moreira; Barreiro, Eliezer J.
PUB. DATE
January 2005
SOURCE
Current Medicinal Chemistry;2005, Vol. 12 Issue 1, p23
SOURCE TYPE
Academic Journal
DOC. TYPE
Article
ABSTRACT
This review aim to demonstrate the role of bioisosterism in rational drug design as well as in the molecular modification and optimization process aiming to improve pharmacodynamic and pharmacokinetic properties of lead compounds.
ACCESSION #
15594299

 

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